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EXP002491

Paper

Delivery System Targeting Hemagglutinin of Influenza Virus A to Facilitate Antisense-Based Anti-H1N1 Therapy (2017)

Peptide

HA-binding peptide HABP / H17

Sequence: SHGRITFAYFAN

RNA

ASO

All experiment fields

Experiment Id EXP002491
Paper Delivery System Targeting Hemagglutinin of Influenza Virus A to Facilitate Antisense-Based Anti-H1N1
Peptide HA-binding peptide HABP / H17
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration Not clearly specified for in vitro assay; plaque assay after IAV-infected A549 cells treated with FT-HABP for 12 h
Mixing Ratio
Formulation Format Covalent peptide-ODN conjugate
Formulation Components HABP peptide + anti-IAV flutide ODN via EMCS linker
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells A549 cells infected with influenza A/FM/1/86 (H1N1)
Animal Model
Administration Route
Output Type Antiviral functional effect / plaque assay
Output Value Plaque formation inhibited more strongly by FT-HABP than unconjugated FT; ~75% inhibition reported in abstract; higher inhibitory effect than ODN alone in Figure 4A
Output Units
Output Notes FITC-HABP colocalized with Cy3-IAV in A549 cells; FT-HABP reduced viral replication in vitro. In vitro effect does not qualify as delivery_success_class=1.
Toxicity Notes No specific toxicity issue reported for FT-HABP in the curated assay.
Curation Notes