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EXP002528

Paper

Introducing a Single-Point Modification to the Cell-Penetrating Peptide PepFect14 Analogue Sequence for Optimising Oligonucleotide Delivery (2025)

Peptide

Met10

Sequence: Stearoyl-AGYLLGKLLMKLAAAALKKLL-NH2

RNA

siRNA

All experiment fields

Experiment Id EXP002528
Paper Introducing a Single-Point Modification to the Cell-Penetrating Peptide PepFect14 Analogue Sequence
Peptide Met10
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed no
Label Confidence medium
In Vitro Functional Effect no
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration 25 nM final siRNA concentration in cell media
Mixing Ratio CPP/siRNA MR20:1 used for main reporter knockdown comparison
Formulation Format noncovalent CPP/siRNA nanoparticle
Formulation Components Met10 CPP self-assembled with luciferase siRNA in ultrapure water after peptide dilution from 10% DMSO/90% ethanol stock.
Size Nm 120.40
Zeta Mv -24.90
Model Scope in_vitro
Model Type in vitro reporter-gene knockdown
Cell Lines Or Primary Cells U87 MG-luc2 human glioma cells stably expressing firefly luciferase
Animal Model
Administration Route in vitro transfection
Output Type luciferase reporter knockdown
Output Value no clear productive siRNA delivery in summary/narrative
Output Units
Output Notes Conservatively labeled inactive/inefficient for siRNA delivery because Met10 was reported as inefficient for NP formation and delivery.
Toxicity Notes No dedicated siRNA-row toxicity flag extracted; overall CPP/RNA nanoparticle study did not emphasize cytotoxicity at tested transfection conditions.
Curation Notes