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EXP002530

Paper

Introducing a Single-Point Modification to the Cell-Penetrating Peptide PepFect14 Analogue Sequence for Optimising Oligonucleotide Delivery (2025)

Peptide

Met10

Sequence: Stearoyl-AGYLLGKLLMKLAAAALKKLL-NH2

RNA

mRNA

All experiment fields

Experiment Id EXP002530
Paper Introducing a Single-Point Modification to the Cell-Penetrating Peptide PepFect14 Analogue Sequence
Peptide Met10
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed no
Label Confidence medium
In Vitro Functional Effect no
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration 80 ng mRNA per well in 96-well plate
Mixing Ratio CPP/mRNA CR2:1 and CR3:1 screened; CR3:1 used for main higher-efficiency comparison
Formulation Format noncovalent CPP/mRNA nanoparticle
Formulation Components Met10 CPP self-assembled with firefly luciferase mRNA in ultrapure water after peptide dilution from 10% DMSO/90% ethanol stock.
Size Nm 120.40
Zeta Mv -24.90
Model Scope in_vitro
Model Type in vitro mRNA reporter-expression assay
Cell Lines Or Primary Cells HaCaT cells
Animal Model
Administration Route in vitro transfection
Output Type mRNA translation / luciferase reporter expression
Output Value inefficient mRNA delivery
Output Units
Output Notes Met10 was reported as inefficient for NP formation and delivery across siRNA, SCO, and mRNA.
Toxicity Notes At CR3:1, mRNA nanoparticles caused no statistically significant reduction in viability in the reported WST8/CCK-type assay.
Curation Notes