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EXP000041

Paper

Pre-administration of PepFect6-microRNA-146a nanocomplexes inhibits inflammatory responses in keratinocytes and in a mouse model of irritant contact dermatitis (2016)

Peptide

PF14 (PepFect14)

Sequence: stearyl-AGYLLGKLLOOLAAAALOOLL-NH2

RNA

miRNA mimic

All experiment fields

Experiment Id EXP000041
Paper Pre-administration of PepFect6-microRNA-146a nanocomplexes inhibits inflammatory responses in kerati
Peptide PF14 (PepFect14)
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio
Formulation Format CPP/miRNA non-covalent nanocomplex
Formulation Components CPP (PF6/PF14/CADY) + miR-146a mimic at 2:1 charge ratio
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells Human primary keratinocytes (normal human epidermal keratinocytes)
Animal Model
Administration Route
Output Type target gene suppression (RT-qPCR) / uptake (Dy547 microscopy)
Output Value Functional miR-146a effect for PF6/PF14; none for CADY
Output Units
Output Notes Functional but less efficient than PF6 in target-gene suppression.
Toxicity Notes
Curation Notes