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EXP000043

Paper

Pre-administration of PepFect6-microRNA-146a nanocomplexes inhibits inflammatory responses in keratinocytes and in a mouse model of irritant contact dermatitis (2016)

Peptide

PF6 (PepFect6)

Sequence: stearyl-AGYLLGK(K(K2(tfq4)))INLKALAALAKKIL-NH2

RNA

miRNA mimic

All experiment fields

Experiment Id EXP000043
Paper Pre-administration of PepFect6-microRNA-146a nanocomplexes inhibits inflammatory responses in kerati
Peptide PF6 (PepFect6)
Delivery Success Class yes
In Vivo Flag yes
Uptake Confirmed yes
Label Confidence
In Vitro Functional Effect
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio
Formulation Format CPP/miRNA non-covalent nanocomplex
Formulation Components CPP (PF6/PF14/CADY) + miR-146a mimic at 2:1 charge ratio
Size Nm
Zeta Mv
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model C57BL/6 mice, irritant contact dermatitis (PMA-induced ear inflammation)
Administration Route Subcutaneous injection into ear (PF6-miR-146a), then topical PMA
Output Type anti-inflammatory phenotype + target gene suppression
Output Value Reduced ear swelling; reduced pro-inflammatory cytokines/chemokines; Irak1/Card10 down
Output Units
Output Notes PF6-miR-146a pre-administration attenuated inflammation vs PF6-control.
Toxicity Notes
Curation Notes