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EXP000062

Paper

Highly efficient delivery of siRNA to a heart transplant model by a novel cell penetrating peptide–dsRNA binding domain (2014)

Peptide

Hph1–Hph1–dsRBD

Sequence: (YARVRRRGPRR)2–dsRBD

RNA

siRNA

All experiment fields

Experiment Id EXP000062
Paper Highly efficient delivery of siRNA to a heart transplant model by a novel cell penetrating peptide–d
Peptide Hph1–Hph1–dsRBD
Delivery Success Class no
In Vivo Flag yes
Uptake Confirmed yes
Label Confidence
In Vitro Functional Effect
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio
Formulation Format CPP–dsRBD/siRNA non-covalent complex (± CaCl2 condensation)
Formulation Components Hph1–Hph1–dsRBD fusion protein + siRNA
Size Nm
Zeta Mv
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model Mouse heart transplantation model (C57BL/6J)
Administration Route Ex vivo graft perfusion with CPP–siRNA complex
Output Type siRNA distribution in heart tissue
Output Value Widespread siRNA distribution throughout grafted heart
Output Units
Output Notes
Toxicity Notes
Curation Notes