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EXP000115

Paper

Albumin Biomimetic Nanocorona Improves Tumor Targeting and Penetration for Synergistic Therapy of Metastatic Breast Cancer (2017)

Peptide

r9-S-S-DOPE

Sequence: RRRRRRRRR (r9)

RNA

siRNA

All experiment fields

Experiment Id EXP000115
Paper Albumin Biomimetic Nanocorona Improves Tumor Targeting and Penetration for Synergistic Therapy of Me
Peptide r9-S-S-DOPE
Delivery Success Class yes
In Vivo Flag yes
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect
Endosomal Escape Evidence yes
Peptide Concentration 0.5 mg siRNA/kg
Rna Concentration 1.0 mg siRNA/kg
Mixing Ratio 9:1 (w/w) CPP:siRNA; HSA 4:1 (w/w)
Formulation Format CPP nanoassembly (r9-S-S-DOPE / DOPE / IR-780) ± HSA
Formulation Components ~130 nm
Size Nm
Zeta Mv 3.00
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model Orthotopic 4T1 breast cancer mouse model
Administration Route IV (tail vein)
Output Type tumor growth inhibition / metastasis prevention
Output Value 83.6% tumor inhibition; 92.2% lung metastasis inhibition
Output Units
Output Notes
Toxicity Notes No significant body weight loss or systemic toxicity
Curation Notes