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EXP000146

Paper

Stimuli-responsive release and efficient siRNA delivery in non-small cell lung cancer by a poly(L-histidine)-based multifunctional nanoplatform (2020)

Peptide

PD (PEG-PSD) coated PLL

Sequence: poly(sulfadimethoxine) peptide-polymer (no PHis)

RNA

siRNA

All experiment fields

Experiment Id EXP000146
Paper Stimuli-responsive release and efficient siRNA delivery in non-small cell lung cancer by a poly(L-hi
Peptide PD (PEG-PSD) coated PLL
Delivery Success Class no
In Vivo Flag yes
Uptake Confirmed no
Label Confidence high
In Vitro Functional Effect
Endosomal Escape Evidence
Peptide Concentration N/P = 4
Rna Concentration 1 mg siRNA/kg
Mixing Ratio PLL:PD:siRNA optimized
Formulation Format PLL/siRNA nanoparticle with polymer coating
Formulation Components ~101 nm
Size Nm
Zeta Mv 5.70
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model A549 xenograft nude mouse
Administration Route IV (tail vein)
Output Type tumor growth inhibition
Output Value Moderate tumor inhibition (<50%)
Output Units
Output Notes
Toxicity Notes No significant systemic toxicity
Curation Notes