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EXP000202

Paper

Anti-Metastatic Effects on Melanoma via Intravenous Administration of Anti-NF-κB siRNA Complexed with Functional Peptide-Modified Nano-Micelles (2020)

Peptide

CH2R4H2C

Sequence: Cys-His-His-Arg-Arg-Arg-Arg-His-His-Cys

RNA

siRNA

All experiment fields

Experiment Id EXP000202
Paper Anti-Metastatic Effects on Melanoma via Intravenous Administration of Anti-NF-κB siRNA Complexed wit
Peptide CH2R4H2C
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio N/P 10
Formulation Format siRelA/MPEG-PCL-CH2R4H2C micelles
Formulation Components ~50 nm
Size Nm
Zeta Mv 5.00
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells B16F10 melanoma cells
Animal Model
Administration Route
Output Type migration suppression / gene silencing
Output Value
Output Units
Output Notes Strong uptake; wound-healing assay shows migration inhibition without cytotoxicity
Toxicity Notes
Curation Notes