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EXP000203

Paper

Anti-Metastatic Effects on Melanoma via Intravenous Administration of Anti-NF-κB siRNA Complexed with Functional Peptide-Modified Nano-Micelles (2020)

Peptide

CH2R4H2C

Sequence: Cys-His-His-Arg-Arg-Arg-Arg-His-His-Cys

RNA

siRNA

All experiment fields

Experiment Id EXP000203
Paper Anti-Metastatic Effects on Melanoma via Intravenous Administration of Anti-NF-κB siRNA Complexed wit
Peptide CH2R4H2C
Delivery Success Class yes
In Vivo Flag yes
Uptake Confirmed no
Label Confidence high
In Vitro Functional Effect
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio N/P 10
Formulation Format siRelA/MPEG-PCL-CH2R4H2C micelles
Formulation Components ~50 nm
Size Nm
Zeta Mv
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model B16F10 lung metastasis (C57BL/6 mice)
Administration Route Intravenous
Output Type metastasis inhibition
Output Value Significant reduction in lung metastatic nodules
Output Units
Output Notes
Toxicity Notes No systemic toxicity; 100% survival
Curation Notes