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EXP000227

Paper

Self-Assembling Lipid–Peptide Hybrid Nanoparticles of Phospholipid–Nonaarginine Conjugates for Enhanced Delivery of Nucleic Acid Therapeutics (2017)

Peptide

Nonaarginine (9R) + Tat

Sequence: GGGRRRRRRRRR (3G9R core); Tat: GRKKRRQRRRPPQ

RNA

siRNA

All experiment fields

Experiment Id EXP000227
Paper Self-Assembling Lipid–Peptide Hybrid Nanoparticles of Phospholipid–Nonaarginine Conjugates for Enhan
Peptide Nonaarginine (9R) + Tat
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence yes
Peptide Concentration N/P = 10
Rna Concentration 0.1–5 µM
Mixing Ratio N/P = 10
Formulation Format lipid–peptide hybrid nanoparticle (T-hNP)
Formulation Components PL9R + siRNA + POPC + cholesterol + PEG-PE ± Tat-PEG-PE
Size Nm 170.00
Zeta Mv 7.00
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells HeLa-GFP; HeLa-Luc; B16F10
Animal Model
Administration Route
Output Type gene knockdown
Output Value ~50% GFP and luciferase knockdown (Tat-dependent kinetics)
Output Units
Output Notes Tat accelerates uptake and early silencing; effect converges over time
Toxicity Notes Low cytotoxicity; improved vs PEI
Curation Notes