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EXP000628

Paper

Tumor microenvironment-activated cancer cell membrane-liposome hybrid nanoparticle-mediated synergistic metabolic therapy and chemotherapy for NSCLC (2021)

Peptide

MMP9-switchable CPP (R9-PVGLIG-EGGEGGEGG)

Sequence: RRRRRRRRR-PVGLIG-EGGEGGEGG

RNA

siRNA

All experiment fields

Experiment Id EXP000628
Paper Tumor microenvironment-activated cancer cell membrane-liposome hybrid nanoparticle-mediated synergis
Peptide MMP9-switchable CPP (R9-PVGLIG-EGGEGGEGG)
Delivery Success Class yes
In Vivo Flag yes
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect
Endosomal Escape Evidence yes
Peptide Concentration
Rna Concentration
Mixing Ratio N/P 4
Formulation Format Hybrid biomimetic nanoparticles (CLip-PC@CO-LC)
Formulation Components Cancer cell membrane + liposome + CPP + LC + siRNA + DTX
Size Nm 193.00
Zeta Mv
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model A549 xenograft nude mice
Administration Route intravenous
Output Type tumor growth inhibition + survival
Output Value ~83.5% tumor inhibition
Output Units
Output Notes Significant tumor suppression and survival benefit
Toxicity Notes No systemic toxicity
Curation Notes