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EXP000699

Paper

WRAP-based nanoparticles for siRNA delivery: a SAR study and a comparison with lipid-based transfection reagents (2021)

Peptide

W5-4L

Sequence: LRLRWWWRLRL

RNA

siRNA

All experiment fields

Experiment Id EXP000699
Paper WRAP-based nanoparticles for siRNA delivery: a SAR study and a comparison with lipid-based transfect
Peptide W5-4L
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect no
Endosomal Escape Evidence
Peptide Concentration R=20 (~200 nM)
Rna Concentration 10–20 nM
Mixing Ratio 20:1 (peptide:siRNA)
Formulation Format CPP-based nanoparticle
Formulation Components W5-4L WRAP peptide + siRNA
Size Nm 80.00
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells U87 glioblastoma (FLuc/NLuc)
Animal Model
Administration Route
Output Type luciferase knockdown
Output Value variable (0–90%) depending on sequence
Output Units
Output Notes SAR study; helix length and Leu doublets critical for activity
Toxicity Notes Low short-term toxicity
Curation Notes