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EXP001061

Paper

Identifying Antisense Oligonucleotides to Disrupt Small RNA Regulated Antibiotic Resistance via a Cell-Free Transcription−Translation Platform (2023)

Peptide

(KFF)3K

Sequence: KFFKFFKFFK

RNA

PNA (antisense to MicF; 12-1)

All experiment fields

Experiment Id EXP001061
Paper Identifying Antisense Oligonucleotides to Disrupt Small RNA Regulated Antibiotic Resistance via a Ce
Peptide (KFF)3K
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed no
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration 6 µM final (reporter & MIC assays); 3 µM tested (no effect reported); also used 3 µM in combo
Rna Concentration 6 µM final (alone); 3 µM final (in combination with 33-22)
Mixing Ratio N/A (covalent conjugate)
Formulation Format CPP-PNA conjugate (covalent); added directly to E. coli cultures / MIC wells
Formulation Components KFFKFFKFFK-O-aatgatgatagc (SI Table S3)
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells Escherichia coli MG1655 (liquid culture reporter assay and MIC assays)
Animal Model
Administration Route
Output Type ompF-sfgfp reporter derepression; MIC (cephalothin) test
Output Value At 6 µM, reporter fluorescence increased to near reporter-only control after 1 h; MIC for cephalothin showed no difference vs scramble (variability noted)
Output Units
Output Notes Authors report 6 µM CPP-PNA 12-1 restored reporter signal but MIC improvement was not observed for cephalothin; also note unexplained increased fluorescence in some controls with 6 µM 12-1.
Toxicity Notes
Curation Notes