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EXP001291

Paper

Attachment of Cell-Binding Ligands to Arginine-Rich Cell-Penetrating Peptides Enables Cytosolic Translocation of Complexed siRNA (2015)

Peptide

scFvCD7-9LR

Sequence: scFvCD7 +RRRRRRRRR

RNA

siRNA

All experiment fields

Experiment Id EXP001291
Paper Attachment of Cell-Binding Ligands to Arginine-Rich Cell-Penetrating Peptides Enables Cytosolic Tran
Peptide scFvCD7-9LR
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration 5 µM (10:1 ratio in Jurkat)
Rna Concentration ~500 nM (100 pmol in 0.2 mL for Jurkat)
Mixing Ratio 10:1 (peptide:siRNA molar)
Formulation Format electrostatic peptide:siRNA complex
Formulation Components scFvCD7-9LR + siRNA (noncovalent complex)
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells Jurkat (human T cell line)
Animal Model
Administration Route in vitro (cell incubation)
Output Type gene knockdown (CD4 mRNA, qPCR)
Output Value 65.6 ± 3.6% CD4 mRNA reduction at 4 h (vs siLuc control)
Output Units
Output Notes Enhanced uptake into Jurkat (MFI 104.6 ± 12.27). Native 9LR and Lipofectamine 2000 failed to knock down CD4 in Jurkat.
Toxicity Notes Not reported.
Curation Notes