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EXP001503

Paper

Therapeutic potential of a cell penetrating peptide (CPP, NP1) mediated siRNA delivery: Evidence in 3D spheroids of colon cancer cells (2020)

Peptide

NP1

Sequence: STR-H16R8 (stearyl-(His)16-(Arg)8)

RNA

siRNA

All experiment fields

Experiment Id EXP001503
Paper Therapeutic potential of a cell penetrating peptide (CPP, NP1) mediated siRNA delivery: Evidence in
Peptide NP1
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration 6 µM
Rna Concentration 100 nM
Mixing Ratio MR 1/60 (siRNA/NP1; N/R≈60)
Formulation Format noncovalent NP1/siRNA complex (nanoparticle)
Formulation Components NP1 + VEGF-A siRNA (electrostatic complex)
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro (2D)
Cell Lines Or Primary Cells HCT 116 human colon cancer cells (2D monolayer)
Animal Model
Administration Route
Output Type Gene knockdown (qRT-PCR, 48 h)
Output Value ~72% VEGF mRNA knockdown
Output Units
Output Notes NP1-VEGF-siRNA complexes reduced VEGF mRNA by ~72% at 48 h in 2D cells (comparable to Lipofectamine 2000).
Toxicity Notes
Curation Notes