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EXP001608

Paper

Lipid nanocapsule functionalization by lipopeptides derived from human papillomavirus type-16 capsid for nucleic acid delivery into cancer cells (2013)

Peptide

L1 (HPV16 capsid-derived)

Sequence: CTSTTAKRKKRKLK

RNA

pDNA

All experiment fields

Experiment Id EXP001608
Paper Lipid nanocapsule functionalization by lipopeptides derived from human papillomavirus type-16 capsid
Peptide L1 (HPV16 capsid-derived)
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence High
In Vitro Functional Effect no
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration 10 µg/mL (plasmid during COS-7 transfection)
Mixing Ratio Complexation tested: 90 ng DNA with 6–300 µg LNC in 20 µL; full complexation at ~240 µg L1-LNC
Formulation Format peptide-functionalized lipid nanocapsule + pDNA complex
Formulation Components Lipid nanocapsules (LNCs; Labrafac® WL1349 core, Solutol® HS15, Lipoïd® S75-3) surface-functionalized via DSPE-PEG2000-peptide (post-insertion method 2)
Size Nm 61.50
Zeta Mv 17.90
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells COS-7 (luciferase assay); uptake of LNC+DNA also shown in U87MG
Animal Model
Administration Route
Output Type luciferase expression (luminescence)
Output Value No detectable luciferase expression (weak/absent transfection vs lipofectamine control)
Output Units
Output Notes L1-LNCs can complex DNA (gel retardation), but did not yield measurable luciferase expression in COS-7.
Toxicity Notes
Curation Notes