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EXP001610

Paper

Lipid nanocapsule functionalization by lipopeptides derived from human papillomavirus type-16 capsid for nucleic acid delivery into cancer cells (2013)

Peptide

L1 (HPV16 capsid-derived)

Sequence: CTSTTAKRKKRKLK

RNA

siRNA

All experiment fields

Experiment Id EXP001610
Paper Lipid nanocapsule functionalization by lipopeptides derived from human papillomavirus type-16 capsid
Peptide L1 (HPV16 capsid-derived)
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence High
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration 25 nM (during cell treatment)
Mixing Ratio Cell treatment: 25 nM siRNA + 100 µg/mL LNCs (2 h, serum-free)
Formulation Format siRNA–L1-LNC complex
Formulation Components Lipid nanocapsules (LNCs; Labrafac® WL1349 core, Solutol® HS15, Lipoïd® S75-3) surface-functionalized via DSPE-PEG2000-peptide (post-insertion method 2)
Size Nm 73.40
Zeta Mv 11.30
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells Caco-2 (CD133 RT-qPCR)
Animal Model
Administration Route
Output Type RT-qPCR (mRNA knockdown)
Output Value Significant CD133 mRNA downregulation vs controls
Output Units
Output Notes L1-LNCs complex siRNA (gel retardation) and mediate CD133 knockdown in Caco-2.
Toxicity Notes
Curation Notes