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EXP001843

Paper

Development of an Efficient Transdermal Delivery System of Small Interfering RNA Using Functional Peptides, Tat and AT-1002 (2011)

Peptide

AT1002 analog (AT-1002)

Sequence: FCIGRLCG

RNA

siRNA

All experiment fields

Experiment Id EXP001843
Paper Development of an Efficient Transdermal Delivery System of Small Interfering RNA Using Functional Pe
Peptide AT1002 analog (AT-1002)
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed no
Label Confidence medium
In Vitro Functional Effect no
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio AT1002:siRNA weight ratio = 80:1 (prepared 30 min at 4°C)
Formulation Format AT1002 + siRNA mixing solution (non-condensing enhancer)
Formulation Components AT1002 mixed with siRelA; evaluated for RNaseA protection (10 ng RNaseA, 37°C, up to 10 h)
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells
Animal Model
Administration Route
Output Type siRNA stability against RNaseA
Output Value AT1002 improves siRNA stability vs naked (partial protection)
Output Units
Output Notes Relative remaining siRNA quantified by fluorescence vs time.
Toxicity Notes
Curation Notes