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EXP002019

Paper

Cell Targeting Peptide Conjugation to siRNA Polyplexes for Effective Gene Silencing in Cardiomyocytes (2012)

Peptide

PCM + Tat

Sequence: PCM: CWLSEAGPVVTVRALRGTGSW; Tat: YGRKKRRQRRR

RNA

siRNA

All experiment fields

Experiment Id EXP002019
Paper Cell Targeting Peptide Conjugation to siRNA Polyplexes for Effective Gene Silencing in Cardiomyocyte
Peptide PCM + Tat
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration siRNA dose 50 nM (0.35 µg/well)
Rna Concentration 50 nM
Mixing Ratio PCM-siRNA : Tat-siRNA = 1:1
Formulation Format siRNA-pDNA/CD polyplex
Formulation Components PCM-siRNA + Tat-siRNA + plasmid DNA + bioreducible polymer (poly(CBA-DAH))
Size Nm 145.00
Zeta Mv 10.00
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells H9C2 cardiomyocytes; NIH 3T3; Huh7; A549
Animal Model
Administration Route
Output Type gene knockdown / reporter expression
Output Value Significant VEGF knockdown; increased GFP expression in cardiomyocytes
Output Units
Output Notes Functional gene silencing and reporter expression shown; enhanced vs non-targeted systems
Toxicity Notes Cell viability >80%; no significant IFN-α induction
Curation Notes