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EXP002055

Paper

Tumor pH-functionalized and charge-tunable nanoparticles for the nucleus/cytoplasm-directed delivery of oxaliplatin and miRNA in head and neck cancer (2022)

Peptide

R-peptide (NLS)

Sequence: RRRRRRRRRK

RNA

All experiment fields

Experiment Id EXP002055
Paper Tumor pH-functionalized and charge-tunable nanoparticles for the nucleus/cytoplasm-directed delivery
Peptide R-peptide (NLS)
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect
Endosomal Escape Evidence yes
Peptide Concentration
Rna Concentration
Mixing Ratio
Formulation Format Lip-TR/Oxa
Formulation Components Liposome + T-peptide + R-peptide + PGA–PEG
Size Nm 143.10
Zeta Mv -37.80
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells SAS (human tongue squamous carcinoma)
Animal Model
Administration Route
Output Type nuclear drug delivery
Output Value Enhanced nuclear localization of oxaliplatin
Output Units
Output Notes Contributes to in vivo efficacy via nuclear targeting of oxaliplatin; not an RNA delivery system
Toxicity Notes Reduced toxicity vs free Oxa
Curation Notes