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EXP002057

Paper

Loading of cocktail siRNAs into extracellular vesicles via TAT-DRBD peptide for the treatment of castration-resistant prostate cancer (2022)

Peptide

3TD peptide (TAT–TAT–TAT–DRBD)

Sequence: YGRKKRRQRRR ×3 + DRBD

RNA

siRNA (cocktail)

All experiment fields

Experiment Id EXP002057
Paper Loading of cocktail siRNAs into extracellular vesicles via TAT-DRBD peptide for the treatment of cas
Peptide 3TD peptide (TAT–TAT–TAT–DRBD)
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration
Mixing Ratio 4:1 (3TD:siRNA theoretical binding)
Formulation Format Engineered extracellular vesicles (EVs)
Formulation Components WPMY-1-derived EVs loaded via 3TD peptide
Size Nm 144.90
Zeta Mv -18.40
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells LNCaP-AI (androgen-independent prostate cancer)
Animal Model
Administration Route
Output Type gene knockdown, apoptosis induction
Output Value qRT-PCR knockdown of 3 genes; AR protein ↓76%; apoptosis ↑
Output Units
Output Notes Robust multi-gene silencing without reported cytotoxicity
Toxicity Notes No significant toxicity reported
Curation Notes