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EXP002185

Paper

A Novel Cell-Penetrating Peptide–VEGF siRNA Complex That Mediates Inhibition of Angiogenesis (2025)

Peptide

Ara27

Sequence: RNQRKTVRCFRCRQAGHWISDCRLKSK

RNA

siRNA

All experiment fields

Experiment Id EXP002185
Paper A Novel Cell-Penetrating Peptide–VEGF siRNA Complex That Mediates Inhibition of Angiogenesis
Peptide Ara27
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration 1 µM
Rna Concentration 50 nM
Mixing Ratio 1:20 (optimal)
Formulation Format CPP/siRNA complex
Formulation Components Ara27 + siVEGF
Size Nm 180.00
Zeta Mv
Model Scope ex_vivo
Model Type in vitro + ex vivo
Cell Lines Or Primary Cells HUVECs
Animal Model Ex vivo mouse aorta ring
Administration Route
Output Type VEGF knockdown; angiogenesis inhibition
Output Value ≈70% VEGF mRNA reduction
Output Units
Output Notes Reduced VEGF signaling, migration, tube formation, and aortic sprouting
Toxicity Notes Low cytotoxicity and no immunotoxicity
Curation Notes