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EXP002253

Paper

Transdermal siRNA delivery by pH-switchable micelles with targeting effect suppress skin melanoma progression (2020)

Peptide

SCP

Sequence: ACTGSTQHQCG

RNA

siRNA

All experiment fields

Experiment Id EXP002253
Paper Transdermal siRNA delivery by pH-switchable micelles with targeting effect suppress skin melanoma pr
Peptide SCP
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed no
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence yes
Peptide Concentration
Rna Concentration
Mixing Ratio SHP:siRNA w/w 2:1, 5:1, 10:1; N/P not specified for transfection assay
Formulation Format pH-switchable cationic micelles (SHP) assembled from SCP-HA-PAE
Formulation Components SCP (ACTGSTQHQCG) + hyaluronic acid (HA, MW 8000) + poly(β-amino ester) (PAE)
Size Nm 170.00
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells HCT116-Luc
Animal Model
Administration Route cell culture (transfection; 6 h exposure; micelles 1 μg/mL)
Output Type reporter knockdown (luciferase assay)
Output Value up to ~62% knockdown at SHP:siRNA = 5:1 (w/w)
Output Units
Output Notes siRNA-luciferase delivered by SHP; luciferase activity normalized by total protein.
Toxicity Notes SHP showed mild cytotoxicity in B16F10 (≈83% viability at 10 μg/mL).
Curation Notes