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EXP002254

Paper

Transdermal siRNA delivery by pH-switchable micelles with targeting effect suppress skin melanoma progression (2020)

Peptide

SCP

Sequence: ACTGSTQHQCG

RNA

siRNA

All experiment fields

Experiment Id EXP002254
Paper Transdermal siRNA delivery by pH-switchable micelles with targeting effect suppress skin melanoma pr
Peptide SCP
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence yes
Peptide Concentration
Rna Concentration
Mixing Ratio SHP/siRNA N/P = 10:1 (used for release & uptake studies); survivin-siRNA loaded SHP
Formulation Format pH-switchable cationic micelles (SHP) assembled from SCP-HA-PAE
Formulation Components SCP (ACTGSTQHQCG) + hyaluronic acid (HA, MW 8000) + poly(β-amino ester) (PAE)
Size Nm 170.00
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells B16F10 (murine melanoma)
Animal Model
Administration Route cell culture
Output Type apoptosis induction (Annexin V/PI; survivin slicing implied)
Output Value ~4-fold higher apoptosis vs naked siRNA or blank micelles (24 h)
Output Units
Output Notes Also showed cellular uptake (FCM/CLSM) and lysosome escape (LysoTracker signal decreases; endosome burst).
Toxicity Notes Blank SHP: ~83% viability retained at 10 μg/mL; low toxicity attributed to degradable components.
Curation Notes