Back to browse

EXP002339

Paper

Mixed Nanosized Polymeric Micelles as Promoter of Doxorubicin and miRNA-34a Co-Delivery Triggered by Dual Stimuli in Tumor Tissue (2016)

Peptide

TATp

Sequence: CYGRKKRRQRRR

RNA

miRNA

All experiment fields

Experiment Id EXP002339
Paper Mixed Nanosized Polymeric Micelles as Promoter of Doxorubicin and miRNA-34a Co-Delivery Triggered by
Peptide TATp
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration component of micelle (5 mol%)
Rna Concentration 100 nM (typical)
Mixing Ratio PEG1k-PE : PEG2k-CLV-Dox : TAT-PEG1k-PE ≈ 90:5:5
Formulation Format polymeric mixed micelle
Formulation Components PEG1k-PE + PEG2k-CLV-Dox + miRNA-34a-S-S-PE + TAT-PEG1k-PE
Size Nm 15.00
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells HT1080; MCF7; 3D HT1080 spheroids
Animal Model
Administration Route cell culture
Output Type gene knockdown + cytotoxicity
Output Value Bcl2 ↓65%, survivin ↓55%, notch1 ↓45%; viability ↓ to ~40%
Output Units
Output Notes Dual MMP2/GSH-triggered release; Tat enhances uptake and escape
Toxicity Notes Low off-target toxicity; serum-compatible
Curation Notes