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EXP002346

Paper

Coated microneedles mediated intradermal delivery of octaarginine/BRAF siRNA nanocomplexes for anti-melanoma treatment (2018)

Peptide

R8

Sequence: RRRRRRRR

RNA

siRNA

All experiment fields

Experiment Id EXP002346
Paper Coated microneedles mediated intradermal delivery of octaarginine/BRAF siRNA nanocomplexes for anti-
Peptide R8
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration N/P ratio 10:1
Rna Concentration 100 nM
Mixing Ratio N/P = 10
Formulation Format CPP/siRNA nanocomplex
Formulation Components R8 + siBraf
Size Nm 353.00
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells A375 melanoma cells
Animal Model
Administration Route cell culture
Output Type gene knockdown + proliferation inhibition
Output Value BRAF mRNA ↓ ~88%; protein ↓ significantly
Output Units
Output Notes Comparable efficacy to PEI; low cytotoxicity
Toxicity Notes Low toxicity compared to PEI
Curation Notes