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EXP002360

Paper

Lipoprotein-biomimetic nanostructure enables tumor-targeted penetration delivery for enhanced photo-gene therapy towards glioma (2022)

Peptide

D4F

Sequence: FAEKFKEAVKDYFAKFWD

RNA

siRNA

All experiment fields

Experiment Id EXP002360
Paper Lipoprotein-biomimetic nanostructure enables tumor-targeted penetration delivery for enhanced photo-
Peptide D4F
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence medium
In Vitro Functional Effect yes
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration 100 nM (siRNA)
Mixing Ratio
Formulation Format HDL-mimetic nanoparticle co-loading ICG + Chol-siRNA
Formulation Components rHDL/siHIF-ICG: PC + D4F + ICG + Chol-siHIF
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells U87 (glioma); bEnd.3 (BBB model)
Animal Model
Administration Route cell culture (± BBB transwell model; ± 808 nm laser)
Output Type in vitro functional effect (HIF-1α pathway)
Output Value Comparator group; functional effect weaker than ptHDL (as reported)
Output Units
Output Notes HDL-mimic built from D4F peptide; cholesterol-siHIF anchored in phospholipid monolayer; ICG in hydrophobic core
Toxicity Notes Negligible dark cytotoxicity in bEnd.3 (reported for formulations)
Curation Notes