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EXP002456

Paper

Tumor Cell Lysate-Based Multifunctional Nanoparticles Facilitate Enhanced mRNA Delivery and Immune Stimulation for Melanoma Gene Therapy (2024)

Peptide

TAT-iRGD

Sequence: CRGDKGPDC-GRKKRRQRRRC

RNA

mRNA

All experiment fields

Experiment Id EXP002456
Paper Tumor Cell Lysate-Based Multifunctional Nanoparticles Facilitate Enhanced mRNA Delivery and Immune S
Peptide TAT-iRGD
Delivery Success Class yes
In Vivo Flag yes
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect
Endosomal Escape Evidence
Peptide Concentration
Rna Concentration 10–12 µg mRNA per dose
Mixing Ratio MLSV/Bim
Formulation Format lipid–polymer nanoparticle
Formulation Components DOTAP + mPEG-PCL + tumor cell lysate + TAT-iRGD
Size Nm 190.00
Zeta Mv 47.80
Model Scope in_vivo
Model Type in vivo
Cell Lines Or Primary Cells
Animal Model B16 melanoma (subcutaneous and lung metastasis), C57 mice
Administration Route intratumoral and intravenous
Output Type tumor suppression / immune activation
Output Value ≈79% tumor growth inhibition (s.c.); ≈63% (lung metastasis)
Output Units
Output Notes Confirmed Bim expression, apoptosis, DC activation
Toxicity Notes No major organ toxicity
Curation Notes