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EXP002547

Paper

Gene Silencing Mediated by siRNA-binding Fusion Proteins Is Attenuated by Double-stranded RNA-binding Domain Structure (2012)

Peptide

PTD-DRBD

Sequence: YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR

RNA

siRNA

All experiment fields

Experiment Id EXP002547
Paper Gene Silencing Mediated by siRNA-binding Fusion Proteins Is Attenuated by Double-stranded RNA-bindin
Peptide PTD-DRBD
Delivery Success Class no
In Vivo Flag no
Uptake Confirmed yes
Label Confidence high
In Vitro Functional Effect yes
Endosomal Escape Evidence yes
Peptide Concentration 0.4–3.0 µM protein
Rna Concentration 50 nM siRNA
Mixing Ratio 20–60:1 protein:siRNA
Formulation Format Protein–siRNA complex
Formulation Components PTD-DRBD fusion protein electrostatically complexed with siRNA
Size Nm
Zeta Mv
Model Scope in_vitro
Model Type in vitro
Cell Lines Or Primary Cells HeLa
Animal Model
Administration Route
Output Type HPRT mRNA knockdown (RT-qPCR)
Output Value ~82% HPRT knockdown (no chloroquine)
Output Units
Output Notes Efficient knockdown; aggregation-mediated uptake; punctate vesicular localization
Toxicity Notes
Curation Notes